Article: Angiopoietin-like protein 4 decreases blood glucose and improves glucose tolerance but induces hyperlipidemia and hepatic steatosis in mice
| Title | Angiopoietin-like protein 4 decreases blood glucose and improves glucose tolerance but induces hyperlipidemia and hepatic steatosis in mice |
|---|---|
| Authors | Xu, A1 Lam, MC1 Chan, KW1 Wang, Y1 Zhang, J1 Boo, RLC1 Xu, JY1 Chen, B1 Chow, WS1 Tso, AWK1 Lam, KSL1 |
| Keywords | Adipokine Diabetes Fatty liver Metabolism |
| Issue Date | 2005 |
| Publisher | National Academy of Sciences. The Journal's web site is located at http://www.pnas.org |
| Citation | Proceedings Of The National Academy Of Sciences Of The United States Of America, 2005, v. 102 n. 17, p. 6086-6091 [How to Cite?] DOI: http://dx.doi.org/10.1073/pnas.0408452102 |
| Abstract | Angiopoietin-like protein 4 (ANGPTL4) is a circulating protein predominantly expressed in adipose tissue and liver. Several recent studies demonstrated that ANGPTL4 is the target gene of peroxisome proliferation activators, the agonists of which are widely used as the antidiabetic and lipid-lowering drugs. Here we provide evidence that ANGPTL4 is a blood-borne hormone directly involved in regulating glucose homeostasis, lipid metabolism, and insulin sensitivity. Adenovirus-mediated expression of ANGPTL4 potently decreased blood glucose and improved glucose tolerance, whereas it induced hyperlipidemia, fatty liver, and hepatomegaly in C57 mice. In db/db diabetic mice, ANGPTL4 treatment reduced hyperglycemia to a normal level, and markedly alleviated glucose intolerance and hyperinsulinemia. Ex vivo studies on primary rat hepatocytes revealed that ANGPTL4 significantly decreased hepatic glucose production and enhanced insulin-mediated inhibition of gluconeogenesis. Serum levels of ANGPTL4 in human subjects inversely correlated with plasma glucose concentrations and HOMA IR, the homeostasis model assessment of insulin resistance. In patients with type 2 diabetes, serum levels of ANGPTL4 were significantly lower than those in healthy subjects, suggesting that the decreased ANGPTL4 could be a causative factor of this disease. These results collectively indicate that ANGPTL4 exerts distinct effects on glucose and lipid metabolism, and that its beneficial effect on glucose homeostasis might be useful for the treatment of diabetes. © 2005 by The National Academy of Sciences of the USA. |
| ISSN | 0027-8424 2011 Impact Factor: 9.681 2011 SCImago Journal Rankings: 1.754 |
| DOI | http://dx.doi.org/10.1073/pnas.0408452102 |
| ISI Accession Number ID | WOS:000228738800036 |
| PubMed Central ID | PMC1087912 |
| References | References in Scopus |
| dc.contributor.author | Xu, A |
|---|---|
| dc.contributor.author | Lam, MC |
| dc.contributor.author | Chan, KW |
| dc.contributor.author | Wang, Y |
| dc.contributor.author | Zhang, J |
| dc.contributor.author | Boo, RLC |
| dc.contributor.author | Xu, JY |
| dc.contributor.author | Chen, B |
| dc.contributor.author | Chow, WS |
| dc.contributor.author | Tso, AWK |
| dc.contributor.author | Lam, KSL |
| dc.date.accessioned | 2008-06-12T06:35:15Z |
| dc.date.available | 2008-06-12T06:35:15Z |
| dc.date.issued | 2005 |
| dc.description.abstract | Angiopoietin-like protein 4 (ANGPTL4) is a circulating protein predominantly expressed in adipose tissue and liver. Several recent studies demonstrated that ANGPTL4 is the target gene of peroxisome proliferation activators, the agonists of which are widely used as the antidiabetic and lipid-lowering drugs. Here we provide evidence that ANGPTL4 is a blood-borne hormone directly involved in regulating glucose homeostasis, lipid metabolism, and insulin sensitivity. Adenovirus-mediated expression of ANGPTL4 potently decreased blood glucose and improved glucose tolerance, whereas it induced hyperlipidemia, fatty liver, and hepatomegaly in C57 mice. In db/db diabetic mice, ANGPTL4 treatment reduced hyperglycemia to a normal level, and markedly alleviated glucose intolerance and hyperinsulinemia. Ex vivo studies on primary rat hepatocytes revealed that ANGPTL4 significantly decreased hepatic glucose production and enhanced insulin-mediated inhibition of gluconeogenesis. Serum levels of ANGPTL4 in human subjects inversely correlated with plasma glucose concentrations and HOMA IR, the homeostasis model assessment of insulin resistance. In patients with type 2 diabetes, serum levels of ANGPTL4 were significantly lower than those in healthy subjects, suggesting that the decreased ANGPTL4 could be a causative factor of this disease. These results collectively indicate that ANGPTL4 exerts distinct effects on glucose and lipid metabolism, and that its beneficial effect on glucose homeostasis might be useful for the treatment of diabetes. © 2005 by The National Academy of Sciences of the USA. |
| dc.description.nature | published_or_final_version |
| dc.format.extent | 388 bytes |
| dc.format.mimetype | text/html |
| dc.identifier.citation | Proceedings Of The National Academy Of Sciences Of The United States Of America, 2005, v. 102 n. 17, p. 6086-6091 [How to Cite?] DOI: http://dx.doi.org/10.1073/pnas.0408452102 |
| dc.identifier.doi | http://dx.doi.org/10.1073/pnas.0408452102 |
| dc.identifier.epage | 6091 |
| dc.identifier.hkuros | 98180 |
| dc.identifier.hkuros | 120053 |
| dc.identifier.isi | WOS:000228738800036 |
| dc.identifier.issn | 0027-8424 2011 Impact Factor: 9.681 2011 SCImago Journal Rankings: 1.754 |
| dc.identifier.issue | 17 |
| dc.identifier.openurl | ![]() |
| dc.identifier.pmcid | PMC1087912 |
| dc.identifier.pmid | 15837923 |
| dc.identifier.scopus | eid_2-s2.0-20944447890 |
| dc.identifier.spage | 6086 |
| dc.identifier.uri | http://hdl.handle.net/10722/49139 |
| dc.identifier.volume | 102 |
| dc.language | eng |
| dc.publisher | National Academy of Sciences. The Journal's web site is located at http://www.pnas.org |
| dc.publisher.place | United States |
| dc.relation.ispartof | Proceedings of the National Academy of Sciences of the United States of America |
| dc.relation.references | References in Scopus |
| dc.rights | National Academy of Sciences Proceedings. Copyright © National Academy of Sciences. |
| dc.rights | Creative Commons: Attribution 3.0 Hong Kong License |
| dc.subject | Adipokine |
| dc.subject | Diabetes |
| dc.subject | Fatty liver |
| dc.subject | Metabolism |
| dc.title | Angiopoietin-like protein 4 decreases blood glucose and improves glucose tolerance but induces hyperlipidemia and hepatic steatosis in mice |
| dc.type | Article |
Author Affiliations
- The University of Hong Kong


