Article: Nuclear penetration of surface functionalized gold nanoparticles
| Title | Nuclear penetration of surface functionalized gold nanoparticles |
|---|---|
| Authors | Gu, YJ2 Cheng, J2 Lin, CC2 Lam, YW2 Cheng, SH2 Wong, WT1 |
| Keywords | Biomaterials Gold nanoparticles Nuclear penetration Surface modification |
| Issue Date | 2009 |
| Publisher | Academic Press. The Journal's web site is located at http://www.elsevier.com/locate/taap |
| Citation | Toxicology And Applied Pharmacology, 2009, v. 237 n. 2, p. 196-204 [How to Cite?] DOI: http://dx.doi.org/10.1016/j.taap.2009.03.009 |
| Abstract | Free gold nanoparticles easily aggregate when the environment conditions change. Here, gold nanoparticles (AuNPs) with average diameter of 3.7 nm were prepared and then modified with poly(ethylene glycol) (PEG) to improve stability. The gold nanoparticles were first surface-modified with 3-mercaptopropionic acid (MPA) to form a self-assembled monolayer and subsequently conjugated with NH2-PEG-NH2 through amidation between the amine end groups on PEG and the carboxylic acid groups on the particles. The biocompatibility and intracellular fate of PEG-modified gold nanoparticles (AuNP@MPA-PEG) were then studied in human cervical cancer (HeLa) cells. Cell viability test showed that AuNP@MPA-PEG did not induce obvious cytotoxicity. Both confocal laser scanning microscopy and transmission electron microscopy demonstrated that AuNP@MPA-PEG entered into mammalian cells and the cellular uptake of AuNP@MPA-PEG was time-dependent. Inductively coupled plasma mass spectrometry and confocal microscopy imaging further demonstrated that AuNP@MPA-PEG penetrated into the nucleus of mammalian cells upon exposure for 24 h. These results suggest that surface modification can enhance the stability and improve the biocompatibility. This study also indicates that AuNP@MPA-PEG can be used as potential nuclear targeted drug delivery carrier. © 2009 Elsevier Inc. All rights reserved. |
| ISSN | 0041-008X 2011 Impact Factor: 4.447 2011 SCImago Journal Rankings: 0.288 |
| DOI | http://dx.doi.org/10.1016/j.taap.2009.03.009 |
| References | References in Scopus |
| dc.contributor.author | Gu, YJ | ||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|
| dc.contributor.author | Cheng, J | ||||||||||
| dc.contributor.author | Lin, CC | ||||||||||
| dc.contributor.author | Lam, YW | ||||||||||
| dc.contributor.author | Cheng, SH | ||||||||||
| dc.contributor.author | Wong, WT | ||||||||||
| dc.date.accessioned | 2010-05-31T03:30:32Z | ||||||||||
| dc.date.available | 2010-05-31T03:30:32Z | ||||||||||
| dc.date.issued | 2009 | ||||||||||
| dc.description.abstract | Free gold nanoparticles easily aggregate when the environment conditions change. Here, gold nanoparticles (AuNPs) with average diameter of 3.7 nm were prepared and then modified with poly(ethylene glycol) (PEG) to improve stability. The gold nanoparticles were first surface-modified with 3-mercaptopropionic acid (MPA) to form a self-assembled monolayer and subsequently conjugated with NH2-PEG-NH2 through amidation between the amine end groups on PEG and the carboxylic acid groups on the particles. The biocompatibility and intracellular fate of PEG-modified gold nanoparticles (AuNP@MPA-PEG) were then studied in human cervical cancer (HeLa) cells. Cell viability test showed that AuNP@MPA-PEG did not induce obvious cytotoxicity. Both confocal laser scanning microscopy and transmission electron microscopy demonstrated that AuNP@MPA-PEG entered into mammalian cells and the cellular uptake of AuNP@MPA-PEG was time-dependent. Inductively coupled plasma mass spectrometry and confocal microscopy imaging further demonstrated that AuNP@MPA-PEG penetrated into the nucleus of mammalian cells upon exposure for 24 h. These results suggest that surface modification can enhance the stability and improve the biocompatibility. This study also indicates that AuNP@MPA-PEG can be used as potential nuclear targeted drug delivery carrier. © 2009 Elsevier Inc. All rights reserved. | ||||||||||
| dc.description.nature | Link_to_subscribed_fulltext | ||||||||||
| dc.identifier.citation | Toxicology And Applied Pharmacology, 2009, v. 237 n. 2, p. 196-204 [How to Cite?] DOI: http://dx.doi.org/10.1016/j.taap.2009.03.009 | ||||||||||
| dc.identifier.doi | http://dx.doi.org/10.1016/j.taap.2009.03.009 | ||||||||||
| dc.identifier.epage | 204 | ||||||||||
| dc.identifier.hkuros | 156628 | ||||||||||
| dc.identifier.isi | WOS:000266289200008
Funding Information: The work described in this paper was totally supported by a grant from the City University of Hong Kong (Project No. CityU 160108). Dr. Gu acknowledges the receipt of post-doctoral fellowship from the City University of Hong Kong Research Enhancement Scheme for their financial support. We also acknowledge the Hong Kong Research Grants Council and The University of Hong Kong for financial support. | ||||||||||
| dc.identifier.issn | 0041-008X 2011 Impact Factor: 4.447 2011 SCImago Journal Rankings: 0.288 | ||||||||||
| dc.identifier.issue | 2 | ||||||||||
| dc.identifier.openurl | ![]() | ||||||||||
| dc.identifier.pmid | 19328820 | ||||||||||
| dc.identifier.scopus | eid_2-s2.0-67349146754 | ||||||||||
| dc.identifier.spage | 196 | ||||||||||
| dc.identifier.uri | http://hdl.handle.net/10722/58451 | ||||||||||
| dc.identifier.volume | 237 | ||||||||||
| dc.language | eng | ||||||||||
| dc.publisher | Academic Press. The Journal's web site is located at http://www.elsevier.com/locate/taap | ||||||||||
| dc.publisher.place | United States | ||||||||||
| dc.relation.ispartof | Toxicology and Applied Pharmacology | ||||||||||
| dc.relation.references | References in Scopus | ||||||||||
| dc.subject | Biomaterials | ||||||||||
| dc.subject | Gold nanoparticles | ||||||||||
| dc.subject | Nuclear penetration | ||||||||||
| dc.subject | Surface modification | ||||||||||
| dc.title | Nuclear penetration of surface functionalized gold nanoparticles | ||||||||||
| dc.type | Article |
Author Affiliations
- The University of Hong Kong
- City University of Hong Kong


