Article: Smad3 mediates cardiac inflammation and fibrosis in angiotensin II-induced hypertensive cardiac remodeling
| Title | Smad3 mediates cardiac inflammation and fibrosis in angiotensin II-induced hypertensive cardiac remodeling |
|---|---|
| Authors | Huang, XR3 Chung, ACK3 Yang, F2 Yue, W2 Deng, C1 Lau, CP2 Tse, HF2 Lan, HY3 |
| Keywords | Angiotensin II Cardiac remodeling Hypertension Smad3 TGF-β |
| Issue Date | 2010 |
| Publisher | Lippincott Williams & Wilkins. The Journal's web site is located at http://hyper.ahajournals.org/ |
| Citation | Hypertension, 2010, v. 55 n. 5, p. 1165-1171 [How to Cite?] DOI: http://dx.doi.org/10.1161/HYPERTENSIONAHA.109.147611 |
| Abstract | Although Smad3 is a key mediator of fibrosis, the functional role of Smad3 in hypertensive cardiovascular disease remains unclear. The present study tested the hypothesis that angiotensin II may activate the transforming growth factor-β/Smad3 pathway to mediate hypertensive cardiac remodeling in Smad3 knockout (KO) and wild-type mice by subcutaneous angiotensin II infusion and in the primary culture of Smad3 KO cardiac fibroblasts. Fourteen days after angiotensin II infusion, both Smad3 KO and wild-type mice developed equal levels of high blood pressure. However, hypertensive cardiac fibrosis and inflammation were developed in Smad3 wild-type but not in Smad3 KO mice. This was demonstrated by the findings that mice lacking Smad3 were protected against a fall in left ventricular ejection fraction (P<0.05), an increase in left ventricular mass (P<0.05), and the development of cardiac fibrosis and inflammation, including upregulation of transforming growth factor-β1, connective tissue growth factor, collagen I/III, α-smooth muscle actin, interleukin 1β, tumor necrosis factor-α, monocyte chemoattractant protein 1, intercellular adhesion molecule 1, and an increase in macrophage and T-cell infiltration in left ventricular tissues (all P<0.01, respectively). Additional studies in vitro also revealed that angiotensin II-induced cardiac fibrosis and inflammation were prevented in Smad3 KO cardiac fibroblasts. Inactivation of both Smad3 and nuclear factor κB/p65 signaling pathways was a key mechanism by which Smad3 KO mice were protected from angiotensin II-mediated hypertensive cardiac remodeling. In conclusion, Smad3 plays an essential role in hypertensive cardiac remodeling. Results from this study suggest that targeting Smad3 may be a novel therapeutic strategy for hypertensive cardiovascular disease. Copyright © 2010 American Heart Association. All rights reserved. |
| Description | link_to_OA_fulltext |
| ISSN | 0194-911X 2011 Impact Factor: 6.207 2011 SCImago Journal Rankings: 0.623 |
| DOI | http://dx.doi.org/10.1161/HYPERTENSIONAHA.109.147611 |
| ISI Accession Number ID | WOS:000276672500019 |
| References | References in Scopus |
| dc.contributor.author | Huang, XR |
|---|---|
| dc.contributor.author | Chung, ACK |
| dc.contributor.author | Yang, F |
| dc.contributor.author | Yue, W |
| dc.contributor.author | Deng, C |
| dc.contributor.author | Lau, CP |
| dc.contributor.author | Tse, HF |
| dc.contributor.author | Lan, HY |
| dc.date.accessioned | 2011-07-27T01:30:12Z |
| dc.date.available | 2011-07-27T01:30:12Z |
| dc.date.issued | 2010 |
| dc.description.abstract | Although Smad3 is a key mediator of fibrosis, the functional role of Smad3 in hypertensive cardiovascular disease remains unclear. The present study tested the hypothesis that angiotensin II may activate the transforming growth factor-β/Smad3 pathway to mediate hypertensive cardiac remodeling in Smad3 knockout (KO) and wild-type mice by subcutaneous angiotensin II infusion and in the primary culture of Smad3 KO cardiac fibroblasts. Fourteen days after angiotensin II infusion, both Smad3 KO and wild-type mice developed equal levels of high blood pressure. However, hypertensive cardiac fibrosis and inflammation were developed in Smad3 wild-type but not in Smad3 KO mice. This was demonstrated by the findings that mice lacking Smad3 were protected against a fall in left ventricular ejection fraction (P<0.05), an increase in left ventricular mass (P<0.05), and the development of cardiac fibrosis and inflammation, including upregulation of transforming growth factor-β1, connective tissue growth factor, collagen I/III, α-smooth muscle actin, interleukin 1β, tumor necrosis factor-α, monocyte chemoattractant protein 1, intercellular adhesion molecule 1, and an increase in macrophage and T-cell infiltration in left ventricular tissues (all P<0.01, respectively). Additional studies in vitro also revealed that angiotensin II-induced cardiac fibrosis and inflammation were prevented in Smad3 KO cardiac fibroblasts. Inactivation of both Smad3 and nuclear factor κB/p65 signaling pathways was a key mechanism by which Smad3 KO mice were protected from angiotensin II-mediated hypertensive cardiac remodeling. In conclusion, Smad3 plays an essential role in hypertensive cardiac remodeling. Results from this study suggest that targeting Smad3 may be a novel therapeutic strategy for hypertensive cardiovascular disease. Copyright © 2010 American Heart Association. All rights reserved. |
| dc.description.nature | Link_to_subscribed_fulltext |
| dc.description | link_to_OA_fulltext |
| dc.identifier.citation | Hypertension, 2010, v. 55 n. 5, p. 1165-1171 [How to Cite?] DOI: http://dx.doi.org/10.1161/HYPERTENSIONAHA.109.147611 |
| dc.identifier.doi | http://dx.doi.org/10.1161/HYPERTENSIONAHA.109.147611 |
| dc.identifier.epage | 1171 |
| dc.identifier.hkuros | 187298 |
| dc.identifier.isi | WOS:000276672500019 |
| dc.identifier.issn | 0194-911X 2011 Impact Factor: 6.207 2011 SCImago Journal Rankings: 0.623 |
| dc.identifier.issue | 5 |
| dc.identifier.pmid | 20231525 |
| dc.identifier.scopus | eid_2-s2.0-77951499390 |
| dc.identifier.spage | 1165 |
| dc.identifier.uri | http://hdl.handle.net/10722/135220 |
| dc.identifier.volume | 55 |
| dc.language | eng |
| dc.publisher | Lippincott Williams & Wilkins. The Journal's web site is located at http://hyper.ahajournals.org/ |
| dc.publisher.place | United States |
| dc.relation.ispartof | Hypertension |
| dc.relation.references | References in Scopus |
| dc.subject.mesh | Angiotensin II - pharmacology |
| dc.subject.mesh | Hypertension - chemically induced - physiopathology |
| dc.subject.mesh | Inflammation - prevention and control |
| dc.subject.mesh | Smad3 Protein - deficiency - genetics - physiology |
| dc.subject.mesh | Ventricular Remodeling - drug effects - genetics - physiology |
| dc.subject | Angiotensin II |
| dc.subject | Cardiac remodeling |
| dc.subject | Hypertension |
| dc.subject | Smad3 |
| dc.subject | TGF-β |
| dc.title | Smad3 mediates cardiac inflammation and fibrosis in angiotensin II-induced hypertensive cardiac remodeling |
| dc.type | Article |
Author Affiliations
- National Institute of Diabetes and Digestive and Kidney Diseases
- The University of Hong Kong
- Chinese University of Hong Kong

