Article: Lipoprotein lipase activator ameliorates the severity of dietary steatohepatitis
| Title | Lipoprotein lipase activator ameliorates the severity of dietary steatohepatitis |
|---|---|
| Authors | Yu, J1 Chu, ESH1 Hui, AY1 Cheung, KF1 Chan, HLY1 Leung, WK1 Farrell, GC2 Sung, JJY1 |
| Keywords | Species Index: Mus |
| Issue Date | 2007 |
| Publisher | Academic Press. The Journal's web site is located at http://www.elsevier.com/wps/find/journaldescription.cws_home/622790/description |
| Citation | Biochemical And Biophysical Research Communications, 2007, v. 356 n. 1, p. 53-59 [How to Cite?] DOI: http://dx.doi.org/10.1016/j.bbrc.2007.02.129 |
| Abstract | Dietary model of steatohepatitis was established by feeding mice a methionine choline deficient (MCD) diet. Mice on MCD or control diet for 3 weeks were treated with or without NO-1886, a newly synthetic lipoprotein lipase (LPL) activator. In a separate experiment, NO-1886 was given after pre-treatment with 3 weeks of MCD diet. NO-1886 significantly reduced MCD-induced inflammation by repressing levels of hepatic lipid peroxides and pro-inflammatory tumor necrosis factor-alpha (TNF-α), interleukin-6 (IL-6), and cyclooxygenase-2 (COX-2). In addition, NO-1886 dampened hepatic steatosis via accelerating fatty acid oxidation caused by enhanced expression of PPARα, cytochrome P450-10 (Cyp4a10), and Acyl-CoA oxidase (ACO). It failed to regulate genes of fatty acid uptake and synthesis pathways. In conclusion, NO-1886 ameliorated and induced regression of experimental steatohepatitis via increasing endogenous LPL activation resulting in suppression on pro-inflammatory factors and reduction of hepatic fatty acids. These findings indicate that NO-1886 is a potential therapeutic agent for steatohepatitis. © 2007 Elsevier Inc. All rights reserved. |
| ISSN | 0006-291X 2011 Impact Factor: 2.484 2011 SCImago Journal Rankings: 0.287 |
| DOI | http://dx.doi.org/10.1016/j.bbrc.2007.02.129 |
| ISI Accession Number ID | WOS:000245419300009 |
| References | References in Scopus |
| dc.contributor.author | Yu, J |
|---|---|
| dc.contributor.author | Chu, ESH |
| dc.contributor.author | Hui, AY |
| dc.contributor.author | Cheung, KF |
| dc.contributor.author | Chan, HLY |
| dc.contributor.author | Leung, WK |
| dc.contributor.author | Farrell, GC |
| dc.contributor.author | Sung, JJY |
| dc.date.accessioned | 2011-04-04T07:57:26Z |
| dc.date.available | 2011-04-04T07:57:26Z |
| dc.date.issued | 2007 |
| dc.description.abstract | Dietary model of steatohepatitis was established by feeding mice a methionine choline deficient (MCD) diet. Mice on MCD or control diet for 3 weeks were treated with or without NO-1886, a newly synthetic lipoprotein lipase (LPL) activator. In a separate experiment, NO-1886 was given after pre-treatment with 3 weeks of MCD diet. NO-1886 significantly reduced MCD-induced inflammation by repressing levels of hepatic lipid peroxides and pro-inflammatory tumor necrosis factor-alpha (TNF-α), interleukin-6 (IL-6), and cyclooxygenase-2 (COX-2). In addition, NO-1886 dampened hepatic steatosis via accelerating fatty acid oxidation caused by enhanced expression of PPARα, cytochrome P450-10 (Cyp4a10), and Acyl-CoA oxidase (ACO). It failed to regulate genes of fatty acid uptake and synthesis pathways. In conclusion, NO-1886 ameliorated and induced regression of experimental steatohepatitis via increasing endogenous LPL activation resulting in suppression on pro-inflammatory factors and reduction of hepatic fatty acids. These findings indicate that NO-1886 is a potential therapeutic agent for steatohepatitis. © 2007 Elsevier Inc. All rights reserved. |
| dc.description.nature | link_to_subscribed_fulltext |
| dc.identifier.citation | Biochemical And Biophysical Research Communications, 2007, v. 356 n. 1, p. 53-59 [How to Cite?] DOI: http://dx.doi.org/10.1016/j.bbrc.2007.02.129 |
| dc.identifier.doi | http://dx.doi.org/10.1016/j.bbrc.2007.02.129 |
| dc.identifier.eissn | 1090-2104 |
| dc.identifier.epage | 59 |
| dc.identifier.isi | WOS:000245419300009 |
| dc.identifier.issn | 0006-291X 2011 Impact Factor: 2.484 2011 SCImago Journal Rankings: 0.287 |
| dc.identifier.issue | 1 |
| dc.identifier.pmid | 17350593 |
| dc.identifier.scopus | eid_2-s2.0-33947172627 |
| dc.identifier.spage | 53 |
| dc.identifier.uri | http://hdl.handle.net/10722/132852 |
| dc.identifier.volume | 356 |
| dc.language | eng |
| dc.publisher | Academic Press. The Journal's web site is located at http://www.elsevier.com/wps/find/journaldescription.cws_home/622790/description |
| dc.publisher.place | United States |
| dc.relation.ispartof | Biochemical and Biophysical Research Communications |
| dc.relation.references | References in Scopus |
| dc.subject.mesh | Animals |
| dc.subject.mesh | Benzamides - administration & dosage - pharmacology |
| dc.subject.mesh | Cholesterol - blood |
| dc.subject.mesh | Choline Deficiency |
| dc.subject.mesh | Cyclooxygenase 2 - genetics - metabolism |
| dc.subject.mesh | Diet - adverse effects |
| dc.subject.mesh | Enzyme Activation - drug effects |
| dc.subject.mesh | Fatty Liver - blood - etiology - prevention & control |
| dc.subject.mesh | Gene Expression - drug effects |
| dc.subject.mesh | Hypolipidemic Agents - administration & dosage - pharmacology |
| dc.subject.mesh | Intercellular Adhesion Molecule-1 - genetics - metabolism |
| dc.subject.mesh | Interleukin-6 - genetics - metabolism |
| dc.subject.mesh | Lipogenesis - genetics |
| dc.subject.mesh | Lipoprotein Lipase - genetics - metabolism |
| dc.subject.mesh | Lipoproteins, HDL - blood |
| dc.subject.mesh | Liver - drug effects - metabolism - pathology |
| dc.subject.mesh | Male |
| dc.subject.mesh | Methionine - deficiency |
| dc.subject.mesh | Mice |
| dc.subject.mesh | Mice, Inbred C57BL |
| dc.subject.mesh | Organophosphorus Compounds - administration & dosage - pharmacology |
| dc.subject.mesh | PPAR gamma - genetics - metabolism |
| dc.subject.mesh | RNA, Messenger - genetics - metabolism |
| dc.subject.mesh | Thiobarbituric Acid Reactive Substances - metabolism |
| dc.subject.mesh | Tumor Necrosis Factor-alpha - genetics - metabolism |
| dc.subject | Species Index: Mus |
| dc.title | Lipoprotein lipase activator ameliorates the severity of dietary steatohepatitis |
| dc.type | Article |
Author Affiliations
- Prince of Wales Hospital Hong Kong
- Australian National University

