Grant: Discovery and Pre-Clinical Evaluation of Promising Metal-Based Anti-Cancer Drug Leads

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Project Title
Discovery and Pre-Clinical Evaluation of Promising Metal-Based Anti-Cancer Drug Leads
 
Principal Investigator Che, Chi Ming (Project coordinator / Principal investigator)
Co-Investigator(s) Poon, Ronnie Tung Ping (Co-Investigator)
Lin, Marie Chia-Mi (Co-Investigator)
Ma, Dik Lung (Co-Investigator)
Sun, Raymond Wai Yin (Deputy project coordinator)
Dr Lau Chi Keung (Co-Investigator)
Vanhoutte, Paul Michel Georges Remi (Co-Investigator)
Siu, Annie Fung Ming (Co-Investigator)
Wang, Yu (Co-Investigator)
Leung, Chung Hang (Co-Investigator)
Professor Lau Tai Chu (Co-Investigator)
Project Code
ITS/134/09FP
 
Funding Year
2009/2010
 
Amount
8999900
 
Panel Physical Sciences
Start Date
01-03-2010
 
Expected Completion
31-08-2012
 
Status
Completed
 
Keywords Metal-Based Anti-Cancer Drug
Grant Type/Funding Scheme Innovation and Technology Support Programme (Tier 2)
Duration
30
 
Publication Specific blocking of CREB/DNA binding by cyclometalated platinum(II) complexes
Publication Organoplatinum(II) complexes with nucleobase motifs as inhibitors of human topoisomerase II catalytic activity
Publication Cyclometalated platinum(ii) complexes as topoisomerase IIα poisons
Publication Osmium(vi) complexes as a new class of potential anti-cancer agents
Publication Luminescent cyclometalated platinum(II) complexes containing N-heterocyclic carbene ligands with potent in vitro and in vivo anti-cancer properties accumulate in cytoplasmic structures of cancer cells
Publication Anticancer gold(i)-phosphine complexes as potent autophagy-inducing agents
Publication Anticancer dirhodium(ii,ii) carboxylates as potent inhibitors of ubiquitin-proteasome system
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